Histone Acetyltransferase Inhibitors

CBP/p300

GCN5/PCAF

TIP60

MOZ/MORF

HBO1

Histone Acetyltransferase Inhibitors & Activators

Product Name	CBP/p300	GCN5/PCAF	TIP60	MOZ/MORF	HBO1	Purity
Curcumin	CBP/p300					98.84%
A-485	CBP/p300					99.87%
C646	CBP/p300					99.78%
SGC-CBP30	CBP/p300					99.83%
WM-3835					HBO1	99.63%
PF-9363				MOZ/MORF		99.64%
Butyrolactone 3		GCN5, IC₅₀: 100 μM				99.31%
NSC 228155	KIX-KID, IC₅₀: 0.36 μM					≥98.0%
Anacardic Acid	p300-HAT, IC₅₀: 8.5 μM	PCAF, IC₅₀: 5 μM				98.86%
MG 149	CBP/p300		TIP60			99.86%
CTB	CBP/p300					99.93%
WM-1119				MOZ/MORF		99.57%
GNE-781	CBP/p300					98.16%
NU9056			TIP60			98.81%
PU139	CREBBP, IC₅₀: 2.49 μM p300, IC₅₀: 5.35 μM	GCN5, IC₅₀: 8.39 μM PCAF, IC₅₀: 9.74 μM				99.14%
NEO2734	CBP/p300					99.63%
Garcinol		GCN5/PCAF				≥99.0%
CPI-1612	CBP/p300					99.74%
TH1834			TIP60			99.60%
CPTH2		GCN5				99.82%
TTK21	CBP/p300					99.39%
PF-CBP1 hydrochloride	CREBBP, IC₅₀: 125 nM EP300, IC₅₀: 363 nM CBP, Kd: .19 μM					99.99%
CTPB	CBP/p300					≥99.0%
YF-2	CBP, EC₅₀: 2.75 μM	GCN5, EC₅₀: 49.31 μM GCN5/PCAF, EC₅₀: 29.04 μM				98.76%
I-CBP112	CBP/p300					98.20%
L002	CBP/p300					99.02%
TH1834 dihydrochloride			TIP60			99.68%
GNE-207	CBP, IC₅₀: 1 nM
CBP/p300-IN-12	CBP/p300, IC₅₀: 166 nM					99.70%
Procyanidin B3	CBP/p300					99.63%
PCAF-IN-2		PCAF, IC₅₀: 5.31 μM				≥98.0%
YF-2 hydrochloride	CBP, EC₅₀: 2.75 μM	GCN5, EC₅₀: 49.31 μM GCN5/PCAF, EC₅₀: 29.04 μM				99.61%
Lys-CoA TFA	p300, IC₅₀: 50-500 nM					99.42%
CBP/p300-IN-10	EP300, IC₅₀: 26 nM CREBBP, IC₅₀: 39 nM					98.69%
NiCur	CBP-HAT, IC₅₀: 0.35 μM					99.11%
Naphthol AS-E	KIX-KID, IC₅₀: 2.26 μM					≥98.0%
Curcumin-d₆	CBP/p300					98.00%
CBP/p300-IN-19 hydrochloride	p300-HAT, IC₅₀: 1.4 μM CBP-HAT, IC₅₀: 2.2 μM	PCAF, IC₅₀: >100 μM
CBP/p300-IN-20	CBP/p300, pIC₅₀: 10.1					98.03%
NSC 694623		PCAF, IC₅₀: 15.9 μM				99.36%
DS17701585	EP300, IC₅₀: 0.04 μM CBP, IC₅₀: 0.15 μM
CPTH2 hydrochloride		GCN5
Ep300/CREBBP-IN-2	EP300, IC₅₀: 0.052 μM CREBBP, IC₅₀: 0.148 μM
Ep300/CREBBP-IN-4	EP300, IC₅₀: 0.024 μM CREBBP, IC₅₀: 0.064 μM
CBP/p300-IN-19	p300-HAT, IC₅₀: 1.4 μM CBP-HAT, IC₅₀: 2.2 μM	PCAF, IC₅₀: >100 μM
CBP/p300-IN-18	EP300, IC₅₀: .056 μM
P300 bromodomain-IN-1	p300, IC₅₀: 49 nM
Ep300/CREBBP-IN-3	EP300, IC₅₀: 0.056 μM CREBBP, IC₅₀: 0.095 μM
CAY10669		PCAF, IC₅₀: 662 μM
Ep300/CREBBP-IN-8	EP300, IC₅₀: 0.014 μM CREBBP, IC₅₀: 0.018 μM
KCN1	p300

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